Inomata et al., Br J Pharmacol 1989
:
In contrast, the inhibitory effect of SUN 1165 ( 1 x 10 ( -5 ) M ) on the peak INa gradually progressed and reached a steady-state level about 2 min after the start of drug-application
Yatani et al., Naunyn Schmiedebergs Arch Pharmacol 1984
:
The effects of SUN 1165 on INa resemble those of lidocaine, although the relative importance of use dependent action versus tonic blockade differs from that of lidocaine